Leelamine, Pyruvate dehydrogenase kinase (PDK) inhibitor (ab120923)
Key features and details
- Pyruvate dehydrogenase kinase (PDK) inhibitor
- CAS Number: 1446-61-3
- Purity: > 98%
- Supplied in ethanol (50 mg/ml)
- Form / State: Liquid
- Source: Synthetic
Overview
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Product name
Leelamine, Pyruvate dehydrogenase kinase (PDK) inhibitor -
Description
Pyruvate dehydrogenase kinase (PDK) inhibitor -
Alternative names
- Dehydroabietylamine
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Biological description
Pyruvate dehydrogenase kinase (PDK) inhibitor (IC50 = 9.5 µM). It has weak affinity for human CB1 and CB2 receptors, exhibiting 20% displacement of [3H]-CP55940 at a concentration of 10 µM.
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Purity
> 98% -
CAS Number
1446-61-3 -
Chemical structure
Properties
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Chemical name
(1R,4aS,10aR)-1,2,3,4,4a,9,10,10a-Octahydro-1,4a-dimethyl-7-(1-methylethyl)-1-phenanthrenemethanamine -
Molecular weight
285.47 -
Molecular formula
C20H31N -
Storage instructions
Store at room temperature. -
Solubility overview
Supplied in ethanol (50 mg/ml) -
Handling
Providing storage is as stated on the product vial and the vial is kept tightly sealed, the product can be stored for up to 6 months. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CC(C)C(C=C1)=CC2=C1[C@]3(C)[C@](CC2)([H])[C@@](CN)(C)CCC3 -
Source
Synthetic
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Research areas
