Pimasertib (AS-703026), MEK1/2 inhibitor (ab235569)
Key features and details
- Selective and potent ATP non-competitive allosteric inhibitor of MEK1/2.
- CAS Number: 1236699-92-5
- Purity: > 98%
DMSO 86 mg/mL (199.44 mM)
Insoluble in water and ethanol
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Pimasertib (AS-703026), MEK1/2 inhibitor -
Description
Selective and potent ATP non-competitive allosteric inhibitor of MEK1/2. -
Alternative names
- AS-703026
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Purity
> 98% -
CAS Number
1236699-92-5 -
Chemical structure
Properties
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Chemical name
N-[(2S)-2,3-dihydroxypropyl]-3-[(2-fluoro-4-iodophenyl)amino]-4-pyridinecarboxamide
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Molecular weight
431.20 -
Molecular formula
C15H15FlN3O3 -
PubChem identifier
44187362 -
Storage instructions
Shipped at 4°C. Store at +4°C short term (1-2 weeks). Store at -20°C long term. It is important to note that this is air sensitive and impurities can occur as a result of air oxidation. Store In the Dark. Store under desiccating conditions. -
Solubility overview
DMSO 86 mg/mL (199.44 mM)
Insoluble in water and ethanol
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SMILES
C1=CC(=C(C=C1I)F)NC2=C(C=CN=C2)C(=O)NCC(CO)O -
Source
Synthetic
