Ketanserin tartrate, 5-HT2 antagonist (ab120132)
Key features and details
- Selective 5-HT2 antagonist
- CAS Number: 83846-83-7
- Purity: > 98%
- Soluble in DMSO to 100 mM and in water to 10 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Ketanserin tartrate, 5-HT2 antagonist -
Description
Selective 5-HT2 antagonist -
Biological description
5-HT2A antagonist. Also shows moderate affinity and selectivity for human 5-HT1Dα over 5-HT1β, and affinity at α1 adrenoceptors. Antihypertensive in vivo.
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Purity
> 98% -
CAS Number
83846-83-7 -
Chemical structure
Properties
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Chemical name
3-(2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl)-2,4(1H,3H)-quinazolinedione tartrate -
Molecular weight
545.51 -
Molecular formula
C22H22FN3O3.C4H6O6 -
PubChem identifier
135348 -
Storage instructions
Store at Room Temperature. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 100 mM and in water to 10 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
O=C(O)C(O)C(O)C(=O)O.Fc1ccc(cc1)C(=O)C4CCN(CCN2C(=O)c3ccccc3NC2=O)CC4 -
Source
Synthetic
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Research areas