CGP 7930, Positive allosteric modulator of GABAB receptors (ab120492)
Key features and details
- Positive GABAB receptor allosteric modulator
- CAS Number: 57717-80-3
- Purity: > 98%
- Soluble in DMSO to 100 mM and in ethanol to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
CGP 7930, Positive allosteric modulator of GABAB receptors -
Description
Positive GABAB receptor allosteric modulator -
Biological description
Positive GABAB receptor allosteric modulator (EC50 values are 5.37 and 4.60 μM, respectively). Increases receptor agonist affinity and signal transduction efficacy. Also shown to potentiate receptor response to baclofen (ab120325).
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Purity
> 98% -
CAS Number
57717-80-3 -
Chemical structure
Properties
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Chemical name
3,5-Bis(1,1-dimethylethyl)-4-hydroxy-β,β-dimethylbenzenepropanol -
Molecular weight
292.46 -
Molecular formula
C19H32O2 -
PubChem identifier
5024764 -
Storage instructions
Store at Room Temperature. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 100 mM and in ethanol to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CC(C)(C)c1cc(cc(c1O)C(C)(C)C)CC(C)(C)CO -
Source
Synthetic
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Research areas