Amisulpride, D2/D3 receptor antagonist (ab142480)
Key features and details
- Potent, highly selective D2/D3 receptor antagonist
- CAS Number: 71675-85-9
- Purity: > 98%
- Soluble in DMSO to 50 mM and ethanol to 100 mM (with warming)
- Form / State: Solid
- Source: Synthetic
Overview
-
Product name
Amisulpride, D2/D3 receptor antagonist -
Description
Potent, highly selective D2/D3 receptor antagonist -
Biological description
Potent, highly selective D2/D3 receptor antagonist (Ki values are 2.8 and 3.2 nM for D2 and D3 receptors respectively). Shows atypical antipsychotic effects in vivo. Orally active. Shows limbic selectivity. -
Purity
> 98% -
CAS Number
71675-85-9 -
Chemical structure
Properties
-
Chemical name
4-Amino-N-[(1-ethylpyrrolidin-2-yl)methyl]-5-ethylsulfonyl-2-methoxybenzamide -
Molecular weight
369.48 -
Molecular formula
C17H27N3O4S -
PubChem identifier
2159 -
Storage instructions
Store at Room Temperature. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 50 mM and ethanol to 100 mM (with warming) -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
-
SMILES
CCN1CCCC1CNC(=O)C2=CC(=C(C=C2OC)N)S(=O)(=O)CC -
Source
Synthetic
-
Research areas
