SB 243213 dihydrochloride, 5HT2C receptor antagonist (ab141291)
Key features and details
- Potent, selective 5HT2C receptor antagonist
- CAS Number: 200940-23-4
- Purity: > 99%
- Soluble in DMSO to 50 mM and in ethanol to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
SB 243213 dihydrochloride, 5HT2C receptor antagonist -
Description
Potent, selective 5HT2C receptor antagonist -
Biological description
Potent, selective 5-HT2C receptor antagonist (Ki = 1 nM). Neurological agent. Active in vivo and in vitro.
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Purity
> 99% -
CAS Number
200940-23-4 -
Chemical structure
Properties
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Chemical name
2,3-Dihydro-5-methyl-N-[6-[(2-methyl-3-pyridinyl)oxy]-3-pyridinyl]-6-(trifluoromethyl)-1H-indole-1-carboxamide dihydrochloride -
Molecular weight
501.33 -
Molecular formula
C22H19F3N4O2.2HCl -
PubChem identifier
15981450 -
Storage instructions
Store at +4°C. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 50 mM and in ethanol to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
Cl.Cl.Cc4ncccc4Oc1ccc(cn1)NC(=O)N3CCc2cc(C)c(cc23)C(F)(F)F -
Source
Synthetic
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Research areas