PD 168568 dihydrochloride, D4 antagonist (ab120611)
Key features and details
- Potent and selective D4 antagonist
- CAS Number: 210688-56-5
- Purity: > 99%
- Soluble in water to 50 mM and in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
PD 168568 dihydrochloride, D4 antagonist -
Description
Potent and selective D4 antagonist -
Biological description
Potent and selective D4 antagonist (Ki = 8.8 nM at D4, and 1842 nM at D2). Inhibits amphetamine stimulated locomotor activity in vivo; orally active.
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Purity
> 99% -
CAS Number
210688-56-5 -
Chemical structure
Properties
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Chemical name
3-[2-[4-(3,4-dimethylphenyl)-1-piperazinyl]ethyl]-2,3-dihydro-1H-isoindol-1-one dihydrochloride -
Molecular weight
422.40 -
Molecular formula
C22H27N3O.2HCl -
Storage instructions
Store at Room Temperature. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 50 mM and in DMSO to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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Source
Synthetic
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Research areas
