Efaroxan hydrochloride, alpha2 adrenoceptor and Imidazoline I1 receptor antagonist (ab145186)
Key features and details
- Potent, highly selective α2 adrenoceptor and Imidazoline I1 receptor antagonist
- CAS Number: 89197-00-2
- Purity: > 99%
- Soluble in water to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Efaroxan hydrochloride, alpha2 adrenoceptor and Imidazoline I1 receptor antagonist -
Description
Potent, highly selective α2 adrenoceptor and Imidazoline I1 receptor antagonist -
Biological description
Potent, highly selective α2 adrenoceptor and Imidazoline I1 receptor antagonist (pKi values are 7.87, 7.42, 5.74, 7.28 and 2A, α2B, α2C, I1, and I2 receptors respectively). Shows antihyperglycemic effects in vivo. -
Purity
> 99% -
CAS Number
89197-00-2 -
Chemical structure
Properties
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Chemical name
2-(2-Ethyl-3H-1-benzofuran-2-yl)-4,5-dihydro-1H-imidazole hydrochloride -
Molecular weight
252.74 -
Molecular formula
C13H16N2O.HCl -
PubChem identifier
11957548 -
Storage instructions
Store at Room Temperature. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Toxic, refer to SDS for further information.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CCC1(CC2=CC=CC=C2O1)C3=NCCN3.Cl -
Source
Synthetic
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Research areas
