CYN 154806, selective somatostatin receptor 2 (sst2) antagonist (ab141210)
Key features and details
- Potent selective somatostatin receptor 2 (sst2) antagonist
- CAS Number: 183658-72-2
- Purity: > 98%
- Soluble in water
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
CYN 154806, selective somatostatin receptor 2 (sst2) antagonist -
Description
Potent selective somatostatin receptor 2 (sst2) antagonist -
Biological description
Potent selective somatostatin receptor 2 (sst2) antagonist (pIC50 values are 8.58 (sst2), 5.41 (sst1), 6.07 (sst3), 5.76 (sst4) and 6.48 (sst5) for human recombinant somatostatin receptors).
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Purity
> 98% -
CAS Number
183658-72-2 -
Chemical structure
Properties
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Molecular weight
1197.35 -
Molecular formula
C56H68N12O14S2 -
Sequence
FCYWKTCY (Modifications: N-terminal acetyl; C-terminal amide; Phe-1 = 4-Nitro(Phe); Disulfide bonds: 2-7) -
PubChem identifier
16133842 -
Storage instructions
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water -
Handling
This product is supplied in one (or more) pack size which is freeze dried. Therefore the contents may not be readily visible, as they can coat the bottom or walls of the vial. Please see our FAQs and information page for more details on handling.
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one week. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
C[C@H]([C@H]1C(=O)N[C@@H](CSSC[C@H](C(=O)N[C@H](C(=O)N[C@@H](C(=O)N[C@H](C(=O)N1)CCCCN)CC2=CNC3=CC=CC=C32)CC4=CC=C(C=C4)O)NC(=O)[C@H](CC5=CC=C(C=C5)[N+](=O)[O-])NC(=O)C)C(=O)N[C@H](CC6=CC=C(C=C6)O)C(=O)N)O -
Source
Synthetic
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Research areas
