Carvedilol, beta and alpha1 adrenoceptor antagonist (ab120709)
Key features and details
- Potent β and α1 adrenoceptor antagonist
- CAS Number: 72956-09-3
- Purity: > 99%
- Soluble in DMSO to 100 mM and in ethanol to 50 mM (with warming)
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Carvedilol, beta and alpha1 adrenoceptor antagonist -
Description
Potent β and α1 adrenoceptor antagonist -
Biological description
Potent β and α1 adrenoceptor antagonist (Ki values are 0.81, 0.96 and 2.2 nM for β1, β2 and α1 adrenoceptors, respectively). Shows antihypertensive, antioxidant, antiapoptotic, anti-inflammatory and antifibrotic properties.
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Purity
> 99% -
CAS Number
72956-09-3 -
Chemical structure
Properties
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Chemical name
1-(9H-Carbazol-4-yloxy)-3-[[2-(2-methoxyphenoxy)ethyl]amino]-2-propanol -
Molecular weight
406.48 -
Molecular formula
C24H26N2O4 -
Storage instructions
Store at +4°C. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 100 mM and in ethanol to 50 mM (with warming) -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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Source
Synthetic
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Research areas