Astemizole, histamine H1 receptor antagonist and hERG K+ channel blocker (ab144583)
Key features and details
- Potent, selective histamine H1 receptor antagonist and potent hERG K+ channel blocker
- CAS Number: 68844-77-9
- Purity: > 99%
- Soluble in DMSO to 50 mM and in ethanol to 50 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Astemizole, histamine H1 receptor antagonist and hERG K+ channel blocker -
Description
Potent, selective histamine H1 receptor antagonist and potent hERG K+ channel blocker -
Biological description
Potent, selective histamine H1 receptor antagonist (IC50 = 4 nM) and potent hERG K+ channel blocker (IC50 =0.9 nM). Orally active. Antiallergic agent. Active in vivo and in vitro. -
Purity
> 99% -
CAS Number
68844-77-9 -
Chemical structure
