VUF8430 dihydrobromide, H4 receptor agonist (ab141128)
Key features and details
- Potent and high affinity H4 receptor agonist
- CAS Number: 100130-32-3
- Soluble in water to 100 mM and in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
VUF8430 dihydrobromide, H4 receptor agonist -
Description
Potent and high affinity H4 receptor agonist -
Biological description
Potent and high affinity H4 receptor agonist (pKi = 7.5 and pEC50 = 7.3). Additionally shows activity at H3 receptors (pKi = 6.5).
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CAS Number
100130-32-3 -
Chemical structure
Properties
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Chemical name
2-[(Aminoiminomethyl)amino]ethyl carbamimidothioic acid ester hydrobromide -
Molecular weight
323.05 -
Molecular formula
C4H11N5S.2HBr -
Storage instructions
Store at Room Temperature. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 100 mM and in DMSO to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
Br.Br.N=C(N)NCCSC(N)=N -
Source
Synthetic
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Research areas
