VU0119498, M1 muscarinic receptor agonist and pan mAChR M3, M5 PAM (ab141512)
Key features and details
- M1 muscarinic receptor agonist and pan mAChR M3, M5 PAM
- CAS Number: 79183-37-2
- Purity: > 99%
- Soluble in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
VU0119498, M1 muscarinic receptor agonist and pan mAChR M3, M5 PAM -
Description
M1 muscarinic receptor agonist and pan mAChR M3, M5 PAM -
Biological description
M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM). Neuroprotective agent. Active in vitro.
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Purity
> 99% -
CAS Number
79183-37-2 -
Chemical structure
Properties
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Chemical name
1-[(4-Bromophenyl)methyl]-1H-indole-2,3-dione -
Molecular weight
316.15 -
Molecular formula
C15H10BrNO2 -
PubChem identifier
3008304 -
Storage instructions
Store at +4°C. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
Brc1ccc(cc1)CN3c2ccccc2C(=O)C3=O -
Source
Synthetic
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Research areas
