TC-2403 oxalate, alpha4beta2 nAChR selective agonist (ab120557)
Key features and details
- Potent α4β2 nAChR selective agonist
- CAS Number: 252870-46-5
- Purity: > 99%
- Soluble in water to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
TC-2403 oxalate, alpha4beta2 nAChR selective agonist -
Description
Potent α4β2 nAChR selective agonist -
Alternative names
- RJR 2403
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Biological description
High affinity α4β2 nAChR selective agonist (Ki = 26 nM). Selective for CNS nAChR over muscle, ganglionic or enteric ACh receptors (EC50 = 732 nM in rat thalamic synaptosomes).
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Purity
> 99% -
CAS Number
252870-46-5 -
Chemical structure
Properties
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Chemical name
(E)-N-Methyl-4-(3-pyridinyl)-3-buten-1-amine oxalate -
Molecular weight
252.27 -
Molecular formula
C10H14N2.C2H2O4 -
Storage instructions
Store at +4°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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Source
Synthetic
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Research areas
