SP-2509, LSD1 inhibitor (ab254459)
Key features and details
- Potent, selective and reversible histone demethylase LSD1 inhibitor
- CAS Number: 1423715-09-6
- Purity: > 98%
Soluble in DMSO to 50 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
SP-2509, LSD1 inhibitor -
Description
Potent, selective and reversible histone demethylase LSD1 inhibitor -
Alternative names
- HCI-2509
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Biological description
Potent, selective (IC50 = 13 nM) and reversible inhibitor of the histone demethylase LSD1 (KDM1A). No activity against MAO-A, MAO-B, lactate dehydrogenase and glucose oxidase.
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Purity
> 98% -
General notes
Solutions in DMSO may be stored at -20°C for up to 3 months.
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CAS Number
1423715-09-6 -
Chemical structure
Properties
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Chemical name
N-[(E)-1-(5-Chloro-2-hydroxyphenyl)ethylideneamino]-3-morpholin-4-ylsulfonylbenzamide
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Molecular weight
437.90 -
Molecular formula
C19H20ClN3O5S -
PubChem identifier
135743577 -
Storage instructions
Shipped at Room Temperature. Store at Room Temperature. Store at -20°C long term. Please see notes section. -
Solubility overview
Soluble in DMSO to 50 mM
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Handling
Refer to SDS for further information.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
C/C(=N\NC(=O)C1=CC(=CC=C1)S(=O)(=O)N2CCOCC2)/C3=C(C=CC(=C3)Cl)O -
Source
Synthetic
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Research areas
