SCH-202676, GPCR allosteric modulator (ab144579)
Key features and details
- Non-selective GPCR allosteric modulator
- CAS Number: 70375-43-8
- Purity: > 98%
- Soluble in DMSO to 25 mM (with warming)
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
SCH-202676, GPCR allosteric modulator -
Description
Non-selective GPCR allosteric modulator -
Biological description
Non-selective GPCR allosteric modulator. Inhibits adenosine, opioid, muscarinic, adrenergic and dopaminergic receptors (IC50 values are 0.1-1.8 μM). Inhibits agonist and antagonist binding to GPCRs. -
Purity
> 98% -
CAS Number
70375-43-8 -
Chemical structure
Properties
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Chemical name
N-(2,3-Diphenyl-1,2,4-thiadiazol-5-(2H)-ylidene)methanamine hydrobromide -
Molecular weight
348.26 -
Molecular formula
C15H13N3S.HBr -
PubChem identifier
11957689 -
Storage instructions
Store at Room Temperature. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 25 mM (with warming) -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CN=C1N=C(N(S1)C2=CC=CC=C2)C3=CC=CC=C3.Br -
Source
Synthetic
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Research areas
