LY 225910, CCK2 receptor antagonist (ab141320)
Key features and details
- Potent, selective CCK2 receptor antagonist
- CAS Number: 133040-77-4
- Purity: > 99%
- Soluble in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
LY 225910, CCK2 receptor antagonist -
Description
Potent, selective CCK2 receptor antagonist -
Biological description
Potent, selective CCK2 receptor antagonist (IC50 = 9.3 nM). Shows anxiolytic effects in vivo.
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Purity
> 99% -
CAS Number
133040-77-4 -
Chemical structure
Properties
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Chemical name
2-[2-(5-Bromo-1H-indol-3-yl)ethyl]-3-[3-(1-methylethoxyphenyl]-4(3H)-quinazolinone -
Molecular weight
502.41 -
Molecular formula
C27H24BrN3O2 -
PubChem identifier
4355450 -
Storage instructions
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CC(C)Oc1cccc(c1)N3C(=Nc2ccccc2C3=O)CCc5cnc4ccc(Br)cc45 -
Source
Synthetic
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Research areas
