HTMT (Histamine trifluoromethyl toluidide) dimaleate, H1/H2 receptor agonist (ab141127)
Key features and details
- H1/H2 receptor agonist. More potent than histamine.
- CAS Number: 195867-54-0
- Purity: > 99%
- Soluble in water to 100 mM and in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
HTMT (Histamine trifluoromethyl toluidide) dimaleate, H1/H2 receptor agonist -
Description
H1/H2 receptor agonist. More potent than histamine. -
Biological description
H1/H2 receptor agonist (Ki = 1.2 µM). More potent than histamine (ab120734). Activates IP3/Ca2+ signaling and induces proliferation of small cholangiocytes. Active in vivo.
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Purity
> 99% -
CAS Number
195867-54-0 -
Chemical structure
Properties
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Chemical name
6-[[2-(1H-Imidazol-5-yl)ethyl]amino]-N-[4-(trifluoromethyl)phenyl]heptanamide dimaleate -
Molecular weight
614.57 -
Molecular formula
C19H25F3N4O.2C4H4O4 -
PubChem identifier
57357684 -
Storage instructions
Store at Room Temperature. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 100 mM and in DMSO to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
O=C(O)\C=C/C(=O)O.O=C(O)\C=C/C(=O)O.FC(F)(F)c1ccc(cc1)NC(=O)CCCCC(C)NCCc2cncn2 -
Source
Synthetic
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Research areas
