Droloxifene citrate, estrogen receptor antagonist (ab142745)
Key features and details
- Estrogen receptor antagonist
- CAS Number: 97752-20-0
- Purity: > 98%
- Soluble in ethanol
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Droloxifene citrate, estrogen receptor antagonist -
Description
Estrogen receptor antagonist -
Biological description
Estrogen receptor antagonist. 10-fold greater binding affinity to the estrogen receptor than tamoxifen (ab120656). Inhibits growth of ER-positive tumor cells. Orally active. Antitumor agent. Active in vitro and in vivo. -
Purity
> 98% -
CAS Number
97752-20-0 -
Chemical structure
Properties
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Chemical name
3-[(E)-1-[4-[2-(Dimethylamino)ethoxy]phenyl]-2-phenylbut-1-enyl]phenol citrate -
Molecular weight
579.64 -
Molecular formula
C26H29NO2.C6H8O7 -
PubChem identifier
3033766 -
Storage instructions
Store at Room Temperature. The product can be stored for up to 12 months. -
Solubility overview
Soluble in ethanol -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CCC(=C(C1=CC=C(C=C1)OCCN(C)C)C2=CC(=CC=C2)O)C3=CC=CC=C3.C(C(=O)O)C(CC(=O)O)(C(=O)O)O -
Source
Synthetic
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Research areas
