Capsazepine, TRPV1 antagonist (ab120025)
Key features and details
- TRPV1 antagonist
- CAS Number: 138977-28-3
- Purity: > 98%
- Soluble in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Capsazepine, TRPV1 antagonist -
Description
TRPV1 antagonist -
Biological description
TRPV1 vanilloid receptor antagonist (IC50 = 562 nM). Analgesic in vivo.
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Purity
> 98% -
CAS Number
138977-28-3 -
Chemical structure
Properties
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Chemical name
N-[2-(4-Chlorophenyl)ethyl]-1,3,4,5-tetrahydro-7,8-dihydroxy-2H-2-benzazepine-2-carbothioamide -
Molecular weight
376.90 -
Molecular formula
C19H21ClN2O2S -
PubChem identifier
2733484 -
Storage instructions
Store at +4°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
Clc1ccc(cc1)CCNC(=S)N2Cc3cc(O)c(O)cc3CCC2 -
Source
Synthetic
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Research areas
