BRL 44408 maleate, alpha2A adrenoceptor antagonist (ab120806)
Key features and details
- Selective α2A adrenoceptor antagonist
- CAS Number: 681806-46-2
- Purity: > 99%
- Soluble in water to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
BRL 44408 maleate, alpha2A adrenoceptor antagonist -
Description
Selective α2A adrenoceptor antagonist -
Biological description
Selective α2A adrenoceptor antagonist (Ki values are 5.68 and 651 nM for α2A and α2B, respectively). Centrally active following subcutaneous administration. Demonstrates antidepressant and analgesic activity.
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Purity
> 99% -
CAS Number
681806-46-2 -
Chemical structure
Properties
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Chemical name
2-[(4,5-Dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole maleate -
Molecular weight
331.37 -
Molecular formula
C13H17N3.C4H4O4 -
Storage instructions
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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Source
Synthetic
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Research areas
