Biperiden hydrochloride, M1 receptor antagonist (ab141781)
Key features and details
- Potent, selective M1 receptor antagonist
- CAS Number: 1235-82-1
- Purity: > 99%
- Soluble in water to 5 mM and in DMSO to 10 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Biperiden hydrochloride, M1 receptor antagonist -
Description
Potent, selective M1 receptor antagonist -
Biological description
Potent, selective M1 receptor antagonist (Ki values are 0.48, 2.4, 3.9, 6.3 and 6.3 nM for M1, M4, M3, M2 and M5 receptors respectively). Shows antiparkinsonian effects and induces impairment of cognitive function in vivo. Orally active. -
Purity
> 99% -
CAS Number
1235-82-1 -
Chemical structure
Properties
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Chemical name
1-(5-Bicyclo[2.2.1]hept-2-enyl)-1-phenyl-3-piperidin-1-ylpropan-1-ol hydrochloride -
Molecular weight
347.92 -
Molecular formula
C21H29NO.HCl -
PubChem identifier
92151 -
Storage instructions
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 5 mM and in DMSO to 10 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
C1CCN(CC1)CCC(C2CC3CC2C=C3)(C4=CC=CC=C4)O.Cl -
Source
Synthetic
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Research areas