VU 0240551, KCC2 inhibitor (ab254523)
Key features and details
- K-Cl co-transporter KCC2 inhibitor
- CAS Number: 893990-34-6
Soluble in DMSO up to 100mM and in ethanol to 25mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
VU 0240551, KCC2 inhibitor -
Description
K-Cl co-transporter KCC2 inhibitor -
Alternative names
- CID-7211972
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Biological description
K-Cl co-transporter KCC2 inhibitor (IC50 = 560 nM for K+ uptake assay in KCC2-overexpressing cells). Also inhibits hERG and L-type Ca2+ channels.
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CAS Number
893990-34-6 -
Chemical structure
Properties
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Chemical name
N-(4-Methyl-1,3-thiazol-2-yl)-2-(6-phenylpyridazin-3-yl)sulfanylacetamide
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Molecular weight
342.43 -
Molecular formula
C16H14N4OS2 -
PubChem identifier
7211972 -
Storage instructions
Shipped at Room Temperature. Store at +4°C. -
Solubility overview
Soluble in DMSO up to 100mM and in ethanol to 25mM
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Handling
Refer to SDS for further information.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CC1=CSC(=N1)NC(=O)CSC2=NN=C(C=C2)C3=CC=CC=C3 -
Source
Synthetic
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Research areas