Tolperisone hydrochloride, voltage-gated Na+ and Ca2+ channel blocker (ab141886)
Key features and details
- Voltage-gated Na+ and Ca2+ channel blocker. Antispastic agent.
- CAS Number: 3644-61-9
- Purity: > 98%
- Soluble in water to 50 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Tolperisone hydrochloride, voltage-gated Na+ and Ca2+ channel blocker -
Description
Voltage-gated Na+ and Ca2+ channel blocker. Antispastic agent. -
Biological description
Voltage-gated Na+ and Ca2+ channel blocker. Antispastic agent. Centrally acting muscle relaxant (IC50 = 50 μM, peak-to-peak amplitude of monosynaptic compound action potential). Shows analgesic and anticonvulsant effects in vivo. Orally active. -
Purity
> 98% -
CAS Number
3644-61-9 -
Chemical structure
Properties
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Chemical name
2-Methyl-1-(4-methylphenyl)-3-piperidin-1-ylpropan-1-one hydrochloride -
Molecular weight
281.82 -
Molecular formula
C16H23NO.HCl -
PubChem identifier
92965 -
Storage instructions
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 50 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CC1=CC=C(C=C1)C(=O)C(C)CN2CCCCC2.Cl -
Source
Synthetic
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Research areas
