Sulfaphenazole, CYP2C9 inhibitor (ab145038)
Key features and details
- Selective CYP2C9 inhibitor.
- CAS Number: 526-08-9
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Sulfaphenazole, CYP2C9 inhibitor -
Description
Selective CYP2C9 inhibitor. -
Alternative names
- 2-Phenyl-3-sulfanilamidopyrazole
- 3-(p-Aminobenzenesulfonamido)-2-phenylpyrazole
- 4-Amino-N-(1-phenyl-1H-pyrazol-5-yl)benzenesulfonamide
see all -
Biological description
Selective, competitive CYP2C9 inhibitor (Ki = 0.3 µM). Blocks pro-inflammatory and atherogenic effects of linoleic acid (increase in oxidative stress and activation of AP-1) mediated by CYP2C9. Inhibits bradykinin-induced tPA release. Sulfonamide antibacterial.
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CAS Number
526-08-9 -
Chemical structure
Properties
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Chemical name
4-Amino-N-(1-phenyl-1H-pyrazol-5-yl)benzenesulfonamide -
Molecular weight
314.36 -
Molecular formula
C15H14N4O2S -
Storage instructions
Store at Room Temperature. The product can be stored for up to 12 months. -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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Source
Synthetic
