Mepyramine maleate, H1 inverse agonist (ab120735)
Key features and details
- Selective H1 inverse agonist
- CAS Number: 59-33-6
- Purity: > 99%
- Soluble in water to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Mepyramine maleate, H1 inverse agonist -
Description
Selective H1 inverse agonist -
Alternative names
- Pyrilamine maleate
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Biological description
Selective H1 receptor inverse agonist (Ki = 0.4 nM). Blood-brain barrier permeable. Shows antihistaminergic action. Additionally, inhibits histamine-induced inositol phosphate production and intracellular calcium mobilization.
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Purity
> 99% -
CAS Number
59-33-6 -
Chemical structure
Properties
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Chemical name
N-(4- Methoxyphenyl) methyl- N′,N′-dimethyl-N-(2-pyridinyl)-1,2-ethanediamine maleate -
Molecular weight
401.46 -
Molecular formula
C17H23N3O.C4H4O4 -
Storage instructions
Store at +4°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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Source
Synthetic
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Research areas
