L-694,247, 5-HT1D/5-HT1B receptor agonist (ab120515)
Key features and details
- Highly potent 5-HT1D/5-HT1B receptor agonist
- CAS Number: 137403-12-4
- Purity: > 99%
- Soluble in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
L-694,247, 5-HT1D/5-HT1B receptor agonist -
Description
Highly potent 5-HT1D/5-HT1B receptor agonist -
Biological description
Highly potent, selective 5-HT1D/5-HT1B receptor agonist (pIC50 values are 10.03 and 9.08 at 5-HT1D and 5-HT1B receptors, respectively). Induces partial blockade of water intake.
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Purity
> 99% -
CAS Number
137403-12-4 -
Chemical structure
Properties
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Chemical name
2-[5-[3-(4-Methylsulfonylamino)benzyl-1,2,4-oxadiazol-5-yl]-1H-indol-3-yl]ethanamine -
Molecular weight
411.48 -
Molecular formula
C20H21N5O3S -
Storage instructions
Store at +4°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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Source
Synthetic
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Research areas
