Inhibitor 6e (PRMT1 inhibitor 6e), PRMT1 inhibitor (ab144665)
Key features and details
- PRMT1 inhibitor
- CAS Number: 1025948-98-4
- Purity: > 98%
- Soluble in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Inhibitor 6e (PRMT1 inhibitor 6e), PRMT1 inhibitor -
Description
PRMT1 inhibitor -
Biological description
PRMT1 inhibitor (IC50 values are 4.8 μM and 22 for hPRMT1 and RmtA, respectively). Docks in both binding sites of the histone arginine methyltransferase pocket.
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Purity
> 98% -
CAS Number
1025948-98-4 -
Chemical structure
Properties
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Chemical name
4-Amino-3,5-dibromo-2-(2,4,5,7-tetrabromo-6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid -
Molecular weight
820.70 -
Molecular formula
C20H7Br6NO5 -
PubChem identifier
16116049 -
Storage instructions
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
O=C(O)c4cc(Br)c(N)c(Br)c4C=2c3cc(Br)c(O)c(Br)c3OC=1C=2C=C(Br)C(=O)C=1Br -
Source
Synthetic
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Research areas
