Harmine, DYRK1A inhibitor (ab120225)
Key features and details
- Potent and selective inhibitor of DYRK1A
- CAS Number: 442-51-3
- Purity: > 98%
- Soluble in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Harmine, DYRK1A inhibitor -
Description
Potent and selective inhibitor of DYRK1A -
Biological description
Potent and selective inhibitor of DYRK1A (dual specificity tyrosine-phosphorylated and -regulated kinase). (IC50 values are 0.08 (DYRK1A), 0.9 (DYRK2), 0.8 (DYRK3), 4.3 (PIM3) and 1.5 μM (CK1)). 5-HT antagonist and MAO inhibitor. Regulator of PPARγ expression and antidiabetic.
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Purity
> 98% -
CAS Number
442-51-3 -
Chemical structure
