Esmolol, beta1 receptor antagonist (ab146018)
Key features and details
- Short-acting cardioselective β1 receptor antagonist. Antiarrhythmic agent.
- CAS Number: 81147-92-4
- Purity: > 98%
- Soluble in water to 25 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Esmolol, beta1 receptor antagonist -
Description
Short-acting cardioselective β1 receptor antagonist. Antiarrhythmic agent. -
Alternative names
- Beta 1 receptor antagonist
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Biological description
Short-acting cardioselective β1 receptor antagonist. Antiarrhythmic agent. Reversibly inhibits Na+ inward currents (IC50 = 74 μM). Shows antihypertensive effects in vivo. Orally active.
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Purity
> 98% -
CAS Number
81147-92-4 -
Chemical structure
Properties
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Chemical name
Methyl 3-[4-(2-hydroxy-3-propan-2-ylamino-propoxy)phenyl]propanoate -
Molecular weight
295.37 -
Molecular formula
C16H25NO4 -
PubChem identifier
59768 -
Storage instructions
Store at +4°C. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 25 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CC(C)NCC(COC1=CC=C(C=C1)CCC(=O)OC)O -
Source
Synthetic
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Research areas