Desformylflustrabromine hydrochloride, alpha4beta2 modulator (ab142815)
Key features and details
- Selective positive allosteric α4β2 modulator
- CAS Number: 951322-11-5
- Purity: > 98%
- Soluble in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Desformylflustrabromine hydrochloride, alpha4beta2 modulator -
Description
Selective positive allosteric α4β2 modulator -
Biological description
Selective positive allosteric nAChR α4β2 modulator (Ki = 3400 nM). Increases whole cell current when co-applied with effective concentrations of ACh. Anti-addictive effects in vivo.
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Purity
> 98% -
CAS Number
951322-11-5 -
Chemical structure
Properties
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Chemical name
6-Bromo-2-(1,1-dimethyl-2-propen-1-yl)-N-methyl-1H-indole-3-ethanamine hydrochloride -
Molecular weight
357.72 -
Molecular formula
C16H21BrN2.HCl -
PubChem identifier
56675778 -
Storage instructions
Store at +4°C. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
Cl.C=CC(C)(C)c2nc1cc(Br)ccc1c2CCNC -
Source
Synthetic
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Research areas
