CID-2011756, PKD inhibitor (ab144601)
Key features and details
- Cell-permeable, specific, ATP-competitive PKD inhibitor
- CAS Number: 638156-11-3
- Purity: > 98%
- Soluble in DMSO to 100 mM and in ethanol to 10 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
CID-2011756, PKD inhibitor -
Description
Cell-permeable, specific, ATP-competitive PKD inhibitor -
Biological description
Cell-permeable, specific, ATP-competitive protein kinase D inhibitor (IC50 values are 0.6, 0.7 and 3.2 μM at PKD2, PKD3 and PKD1 respectively). Antitumor agent. Active in vitro. -
Purity
> 98% -
CAS Number
638156-11-3 -
Chemical structure
Properties
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Chemical name
5-(3-Chlorophenyl)-N-[4-(4-morpholinylmethyl)phenyl]-2-furancarboxamide -
Molecular weight
396.88 -
Molecular formula
C22H21ClN2O3 -
PubChem identifier
2011756 -
Storage instructions
Store at Room Temperature. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 100 mM and in ethanol to 10 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
C1COCCN1CC2=CC=C(C=C2)NC(=O)C3=CC=C(O3)C4=CC(=CC=C4)Cl -
Source
Synthetic
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Research areas
