BRL 52537 hydrochloride, kappa-opioid agonist (ab120669)
Key features and details
- Highly selective, potent κ-opioid agonist
- CAS Number: 112282-24-3
- Purity: > 99%
- Soluble in water to 5 mM and in DMSO to 25 mM (with warming)
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
BRL 52537 hydrochloride, kappa-opioid agonist -
Description
Highly selective, potent κ-opioid agonist -
Biological description
Highly selective and potent κ-opioid agonist (Ki = 0.24 nM). 25 times more potent than morphine. Neuroprotective effects seen in vivo.
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Purity
> 99% -
CAS Number
112282-24-3 -
Chemical structure
Properties
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Chemical name
2-(3,4-Dichlorophenyl)-1-[2-(1-pyrrolidinylmethyl)-1-piperidinyl]ethanone hydrochloride -
Molecular weight
391.77 -
Molecular formula
C18H24Cl2N2O.HCl -
Storage instructions
Store at Room Temperature. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 5 mM and in DMSO to 25 mM (with warming) -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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Source
Synthetic
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Research areas
