Anpirtoline hydrochloride, 5-HT1B receptor agonist (ab146122)
Key features and details
- Potent 5-HT1B receptor agonist
- CAS Number: 99201-87-3
- Purity: > 99%
- Soluble in water to 100 mM and in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Anpirtoline hydrochloride, 5-HT1B receptor agonist -
Description
Potent 5-HT1B receptor agonist -
Biological description
Potent, selective 5-HT1B receptor agonist (Ki values are 28, 150 and 1490 nM for 5-HT1B, 5-HT1A and 5-HT2 receptors, respectively). Shows antidyskinetic effects in vivo. Blood-brain barrier permeable.
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Purity
> 99% -
CAS Number
99201-87-3 -
Chemical structure
Properties
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Chemical name
2-Chloro-6-(4-piperidinylthio)pyridine hydrochloride -
Molecular weight
265.20 -
Molecular formula
C10H13ClN2S.HCl -
PubChem identifier
6917943 -
Storage instructions
Store at +4°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 100 mM and in DMSO to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
C1CNCCC1SC2=NC(=CC=C2)Cl.Cl -
Source
Synthetic
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Research areas
