VU0255035, muscarinic M1 antagonist (ab141424)
Key features and details
- Highly selective, competitive muscarinic M1 antagonist
- CAS Number: 1135243-19-4
- Purity: > 98%
- Soluble in DMSO to 50mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
VU0255035, muscarinic M1 antagonist -
Description
Highly selective, competitive muscarinic M1 antagonist -
Biological description
Highly selective, competitive muscarinic M1 antagonist (Ki = 14.87 nM). 75-fold selectivity over other receptor subtypes for orthosteric site. Blood-brain barrier permeable.
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Purity
> 98% -
CAS Number
1135243-19-4 -
Chemical structure
Properties
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Chemical name
N-[3-Oxo-3-[4-(4-pyridinyl)-1-piperazinyl]propyl]-2,1,3-benzothiadiazole-4-sulfonamide -
Molecular weight
432.51 -
Molecular formula
C18H20N6O3S2 -
PubChem identifier
22247365 -
Storage instructions
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO to 50mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
O=C(CCNS(=O)(=O)c1cccc2nsnc12)N3CCN(CC3)c4ccncc4 -
Source
Synthetic
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Research areas
