Sumanirole maleate, D2 agonist (ab254491)
Key features and details
- Selective high affinity D2 receptor agonist
- CAS Number: 179386-44-8
Soluble in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Sumanirole maleate, D2 agonist -
Description
Selective high affinity D2 receptor agonist -
Biological description
Selective high affinity D2 receptor agonist (EC50 values are between 17 and 75 nM in cell-based assays). Displays >200-fold selectivity for the D2 receptor against other dopamine receptor subtypes (Ki values are 9.0, 1940, >2190 and >7140 for D2, D3, D4 and D1 receptors respectively.
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CAS Number
179386-44-8 -
Chemical structure
Properties
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Chemical name
(10R)-10-(Methylamino)-1,3-diazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one (Z)-but-2-enedioic acid
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Molecular weight
319.32 -
Molecular formula
C15H17N3O5 -
PubChem identifier
9818478 -
Storage instructions
Shipped at 4°C. Store at +4°C. -
Solubility overview
Soluble in DMSO to 100 mM
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Handling
Refer to SDS for further information.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CN[C@@H]1CC2=C3C(=CC=C2)NC(=O)N3C1.C(=C\C(=O)O)\C(=O)O -
Source
Synthetic