Droloxifene, estrogen receptor modulator (ab143610)
Key features and details
- Selective estrogen receptor modulator
- CAS Number: 82413-20-5
- Purity: > 98%
- Soluble in DMSO
- Form / State: Solid
- Source: Synthetic
Overview
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Product name
Droloxifene, estrogen receptor modulator -
Description
Selective estrogen receptor modulator -
Biological description
Selective estrogen receptor modulator. Tamoxifen analog. Induces p53 activation and apoptosis in osteoclasts and MCF-7 cells. Shows tissue selective estrogenic and antiestrogenic effects. Inhibits bone resorption in vivo. Orally active. -
Purity
> 98% -
CAS Number
82413-20-5 -
Chemical structure
Properties
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Chemical name
3-[(E)-1-[4-[2-(Dimethylamino)ethoxy]phenyl]-2-phenylbut-1-enyl]phenol -
Molecular weight
387.51 -
Molecular formula
C26H29NO2 -
PubChem identifier
3033767 -
Storage instructions
Store at Room Temperature. The product can be stored for up to 12 months. -
Solubility overview
Soluble in DMSO -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CCC(=C(C1=CC=C(C=C1)OCCN(C)C)C2=CC(=CC=C2)O)C3=CC=CC=C3 -
Source
Synthetic
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Research areas
