ARC 239 dihydrochloride, alpha2B adrenoceptor antagonist (ab146143)
Key features and details
- Selective α2B adrenoceptor antagonist
- CAS Number: 55974-42-0
- Purity: > 99%
- Soluble in water to 100 mM and in DMSO to 100 mM
- Form / State: Solid
- Source: Synthetic
Overview
-
Product name
ARC 239 dihydrochloride, alpha2B adrenoceptor antagonist -
Description
Selective α2B adrenoceptor antagonist -
Biological description
Selective α2B adrenoceptor antagonist (-log Kb = 8.51). Active in vivo and in vitro.
-
Purity
> 99% -
CAS Number
55974-42-0 -
Chemical structure
Properties
-
Chemical name
2-[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]-4,4-dimethyl-1,3(2H,4H)-isoquinolinedione dihydrochloride -
Molecular weight
480.43 -
Molecular formula
C24H29N3O3.2HCl -
PubChem identifier
10345075 -
Storage instructions
Store at +4°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
Solubility overview
Soluble in water to 100 mM and in DMSO to 100 mM -
Handling
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
-
SMILES
CC1(C2=CC=CC=C2C(=O)N(C1=O)CCN3CCN(CC3)C4=CC=CC=C4OC)C.Cl.Cl -
Source
Synthetic
-
Research areas
